some unusual reactions of 3-phenylaminoisoxazol-5 (2h)- ones

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چکیده

3-phenylaminoisoxazol-5(2h)-ones,s ubstituted on nitrogen with an isoquinoline or quinazoline group, react with tertiary amine bases to give imidazo annelated compounds. when the n-substituent is a nitropyridine, 2-aminoindole derivatives are formed instead. evidence is presented that the reactions proceed by initial addition of the tertiary arnine to c-4

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SOME UNUSUAL REACTIONS OF 3-PHENYLAMINOISOXAZOL-5 (2H)- ONES

3-Phenylaminoisoxazol-5(2H)-ones,s ubstituted on nitrogen with an isoquinoline or quinazoline group, react with tertiary amine bases to give imidazo annelated compounds. When the N-substituent is a nitropyridine, 2-aminoindole derivatives are formed instead. Evidence is presented that the reactions proceed by initial addition of the tertiary arnine to C-4

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عنوان ژورنال:
journal of sciences islamic republic of iran

جلد ۱۱، شماره ۱، صفحات ۰-۰

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